Protease Inhibitors and Phosphatase Inhibitors
MilliporeSigma™ Calbiochem™ Zebularine
A cell-permeable chemically stable cytidine analog that displays antitumor properties.
MilliporeSigma™ Calbiochem™ SB 202190
SB 202190, CAS 152121-30-7, is a potent, reversible, competitive inhibitor of p38. Inhibits p38 phosphorylation of myelin basic protein. Blocks the activity of p38β (K
MilliporeSigma™ Calbiochem™ Brk Inhibitor, Cpd 4f
A cell permeable, highly potent, and very selective inhibitor of breast tumor kinase (Brk; IC50 = 3.15 nM). Displays anti-proliferative activity against multiple breast cancer cell lines.
MilliporeSigma™ Calbiochem™ Cathepsin Inhibitor III
The Cathepsin Inhibitor III controls the biological activity of Cathepsin. This small molecule/inhibitor is primarily used for Protease Inhibitors applications.
MilliporeSigma™ Calbiochem™ Erastin
A cell-permeable piperazinyl-quinazolinone compound that exhibits oncogene-selective lethality.
MilliporeSigma™ Calbiochem™ Sphingosine Kinase Inhibitor
The Sphingosine Kinase Inhibitor, also referenced under CAS 1177741-83-1, controls the biological activity of Sphingosine Kinase. This small molecule/inhibitor is primarily used for Cell Signaling applications.
MilliporeSigma™ Calbiochem™ Caspase-6 Substrate III, Fluorogenic
A fluorogenic substrate for caspase-6 (Mch2).
MilliporeSigma™ Calbiochem™ Autotaxin Inhibitor II, HA130
A thiazolidinedione that is designed to target the ATX active site thr210 with a boronic moiety and shown to potently inhibit ATX lysoPLD activity (IC50 ∽28nM using recombinant human ATX or human plasma) in a reversible manner with a mixed-type Lineweaver-Burk kinet
MilliporeSigma™ Calbiochem™ 1-Oleoyl-2-acetyl-sn-glycerol
Cell-permeable diacylglycerol analog that activates Ca2+-dependent protein kinase C.
MilliporeSigma™ Calbiochem™ 11beta-HSD1 Inhibitor, 10j
The 11beta-HSD1 Inhibitor, 10j, also referenced under CAS 1009373-58-3, controls the biological activity of 11beta-HSD1. This small molecule/inhibitor is primarily used for Protease Inhibitors applications.
MP Biomedicals™ Protease Inhibitor Cocktail Kit
Research Use Only
MilliporeSigma™ Calbiochem™ PK11195
An isoquinoline carboxamide that acts as a potent ligand for peripheral bezodiazepine receptor (Kd = 20
MilliporeSigma™ Calbiochem™ Adipogenesis Inducers Panel
A panel containing eight adipogenesis inducers useful for differentiation of preadipocyte to mature adipocyte.
Aprotinin, Analytical Grade, MP Biomedicals™
Forms stable complexes with enzymes. Aprotinin, Analytical Grade, MP Biomedicals is a competitive serine proteinase inhibitor that works by blocking the active sites of enzymes. This binding is reversible with most aprotinin-protease complexes, dissociati